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| Cat. Number | PD 81723 |
| Chemical Name | PD 81723 |
| CAS Number | [132861-87-1] |
| Mol. Formula | C14H12F3NOS |
| Mol. Weight | 299.31 |
| Qty 1 |
10mg |
| Qty 2 | 50mg |
| Synonym | (2-Amino-4,5-dimethyl-3-thienyl)-[3 -(trifluoromethyl)phenyl]methanone |
| Solubility | Soluble to 100 mM in ethanol and to 100 mM in DMSO |
| Storage condition | Store at RT |
| References | Allosteric potentiator at the adenosine A1 receptor; acts via agonist-dependent and -independent mechanisms. Enhances agonist affinity for, and increased t½ of dissociation from, the receptor. Also inhibits basal and forskolin-stimulated adenylyl cyclase (AC) activity in A1 receptors expressed in CHO cells, possibly via direct potentiation of constitutive receptor activity or by direct inhibition of AC. Active in vivo. Purity: >99 % |




