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/ Products Classification 点击展开+Cat. Number | PD 81723 |
Chemical Name | PD 81723 |
CAS Number | [132861-87-1] |
Mol. Formula | C14H12F3NOS |
Mol. Weight | 299.31 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | (2-Amino-4,5-dimethyl-3-thienyl)-[3 -(trifluoromethyl)phenyl]methanone |
Solubility | Soluble to 100 mM in ethanol and to 100 mM in DMSO |
Storage condition | Store at RT |
References | Allosteric potentiator at the adenosine A1 receptor; acts via agonist-dependent and -independent mechanisms. Enhances agonist affinity for, and increased t½ of dissociation from, the receptor. Also inhibits basal and forskolin-stimulated adenylyl cyclase (AC) activity in A1 receptors expressed in CHO cells, possibly via direct potentiation of constitutive receptor activity or by direct inhibition of AC. Active in vivo. Purity: >99 % |