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/ Products Classification 点击展开+Cat. Number | 287139609265726 |
Chemical Name | AMG 9810 |
CAS Number | [545395-94-6] |
Mol. Formula | C21H23NO3 |
Mol. Weight | 337.42 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | (2E)-N-(2,3-Dihydro-1,4-benzodioxin -6-yl)-3-[4-(1,1-dimethylethyl)phenyl]-2-propenami de |
Solubility | Soluble to 50 mM in DMSO and to 100 mM in ethanol |
Storage condition | Desiccate at +4°C |
References | Potent and selective, competitive vanilloid TRPV1 receptor antagonist (IC50 = 17 nM). Inhibits capsaicin-, proton-, heat- and endogenous ligand-induced activation of human and rat recombinant TRPV1 receptors. Displays antihyperalgesic properties in a rat model of inflammatory pain. Purity: >98 % |