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| Cat. Number | 284420124258071 |
| Chemical Name | BAN ORL 24 |
| CAS Number | [475150-69-7] |
| Mol. Formula | C27H35N3O2.2HCl |
| Mol. Weight | 506.51 |
| Qty 1 |
10mg |
| Qty 2 | 50mg |
| Synonym | (2R)-1-(Phenylmethyl)-N-[3-(spiro[i sobenzofuran-1(3H),4'-piperidin]-1-yl)propyl-2-pyrr olidinecarboxamide |
| Solubility | Soluble to 100 mM in water and to 100 mM in DMSO |
| Storage condition | Desiccate at RT |
| References | Potent and selective NOP receptor antagonist (IC50 values are 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors respectively). Inhibits nociceptin-induced stimulation of [35S]-GTPγS binding and Ca2+ mobilization in CHO cells in vitro and antagonizes NOP agonist-induced reduction in locomotor activity in vivo. Brain penetrant. Purity: >99 % |
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