服务热线
021-60498804
产品中心
/ Products Classification 点击展开+Cat. Number | 282625446989065 |
Chemical Name | CGP 55845 hydrochloride |
CAS Number | [149184-22-5] |
Mol. Formula | C18H22Cl2NO3P.HCl |
Mol. Weight | 438.71 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | (2S)-3-[[(1S)-1-(3,4-Dichlorophenyl )ethyl]amino-2-hydroxypropyl](phenylmethyl)phosphi nic acid hydrochloride |
Solubility | Soluble to 100 mM in DMSO |
Storage condition | Store at RT |
References | Potent, selective GABAB receptor antagonist (IC50 = 5 nM) that prevents agonist binding (pKi = 8.35) and inhibits GABA and glutamate release (pEC50 values are 8.08 and 7.85 respectively). Inhibits GABAB responses to baclofen (IC50 = 130 nM in an isoproterenol assay) and potentiates the hypoglycemic response to glucose in vitro. Purity: >98 % |
下一个:CGP 57380上一个:CGP 54626 hydrochloride |