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/ Products Classification 点击展开+Cat. Number | L-371,257 |
Chemical Name | L-371,257 |
CAS Number | [162042-44-6] |
Mol. Formula | C28H33N3O6 |
Mol. Weight | 507.59 |
Qty 1 |
10mg |
Synonym | 1-[4-[(1-Acetyl-4-piperidinyl)oxy]- 2-methoxybenzoyl]-4-(2-oxo-2H-3,1-benzoxazin-1(4H) -yl)piperidine |
Solubility | Soluble to 100 mM in DMSO and to 100 mM in ethanol |
Storage condition | Store at RT |
References | Potent, high affinity human oxytocin (OT) receptor antagonist (Ki = 4.6 nM) that displays > 800-fold selectivity over human arginine vasopressin receptors V1a and V2. Antagonizes oxytocin-induced contractions in isolated rat uterine tissue (pA2 = 8.44) and in anesthetised rats following intravenous and intraduodenal administration. Orally active. Purity: >99 % |
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