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/ Products Classification 点击展开+Cat. Number | L-368,899 hydrochloride |
Chemical Name | L-368,899 hydrochloride |
CAS Number | [148927-60-0] |
Mol. Formula | C26H42N4O5S2.HCl |
Mol. Weight | 591.23 |
Qty 1 |
1mg |
Qty 2 | 10mg |
Synonym | (2S)-2-Amino-N-[(1S,2S,4R)-7,7-dime thyl-1-[[[4-(2-methylphenyl)-1-piperazinyl]sulfony l]methyl]bicyclo[2.2.1]hept-2-yl]-4-(methylsulfony l)butanamide |
Solubility | Soluble to 100 mM in water and to 100 mM in DMSO |
Storage condition | Store at +4°C |
References | Potent, non-peptide and orally active oxytocin receptor antagonist (IC50 = 8.9 nM) that displays > 40-fold selectivity over vasopressin V1a and V2 receptors (IC50 values are 370 and 570 nM respectively). Antagonizes oxytocin-induced uterine contractions in vitro and in vivo. Purity: >99 % |