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/ Products Classification 点击展开+Cat. Number | Org 27569 |
Chemical Name | Org 27569 |
CAS Number | [868273-06-7] |
Mol. Formula | C24H28ClNO3 |
Mol. Weight | 409.95 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | 5-Chloro-3-ethyl-N-[2-[4-(1-piperid inyl)phenyl]ethyl-1H-indole-2-carboxamide |
Solubility | Soluble to 100 mM in DMSO |
Storage condition | Store at RT |
References | Potent CB1 receptor allosteric modulator (pEC50 = 8.24). Significantly increases binding of the CB1 agonist [3H]CP 55.940 (pKb = 5.67) and decreases binding of the CB1 inverse agonist [3H]SR 141716A (pKb = 5.95). Inhibits CB1 receptor antagonist efficacy in vitro (pKb = 7.57). Purity: >99 % |