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Cat. Number
PF 04217903 mesylate
Chemical Name
PF 04217903 mesylate
CAS Number
[956906-93-7]
Mol. Formula
C19H16N8O.CH3SO3H
Mol. Weight
468.49
Qty 1
10mg
Qty 2
50mg
Synonym
4-[1-(6-Quinolinylmethyl)-1H-1,2,3- triazolo[4,5-b]pyrazin-6-yl]-1H-pyrazole-1-ethanol mesylate
Solubility
Soluble to 100 mM in DMSO
Storage condition
Store at +4°C
References
Highly selective, high affinity c-Met inhibitor (Ki = 6-7 nM against wild type c-Met). Displays >1000-fold selectivity for c-Met over a panel of 208 kinases.
Purity: >98 %
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