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/ Products Classification 点击展开+Cat. Number | RS 39604 hydrochloride |
Chemical Name | RS 39604 hydrochloride |
CAS Number | [167710-87-4] |
Mol. Formula | C26H36ClN3O6S.HCl |
Mol. Weight | 590.56 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | 1-[4-Amino-5-chloro-2-(3,5-dimethox yphenyl)methyloxy]-3-[1-[2-methylsulphonylamino]et hyl]piperidin-4-yl]propan-1-one hydrochloride |
Solubility | Soluble to 100 mM in DMSO |
Storage condition | Store at RT |
References | A potent and selective 5-HT4 antagonist, with a pKi of 9.1 at 5-HT4 receptors in guinea pig striatal membranes and greater than 1000-fold selectivity over 5-HT1A, 2C, 3 and D1, D2, M1, M2, AT1, B1 and α1C receptors. The ketone group gives RS 39604 a relatively long half life; it is also orally active and so suitable for in vivo studies. Purity: >99 % |