您的位置:首页>>糖科学>>Amisulpride
Cat. Number
287204719927263
Chemical Name
Amisulpride
CAS Number
[71675-85-9]
Mol. Formula
C17H27N3O4S
Mol. Weight
369.48
Qty 1
50mg
Synonym
4-Amino-N-[(1-ethyl-2-pyrrolidinyl) methyl]-5-(ethylsulfonyl)-2-benzamide
Solubility
Soluble to 25 mM in 1eq. HCl and to 50 mM in DMSO
Storage condition
Store at -20°C
References
Potent, selective dopamine D2 and D3 receptor antagonist. Ki values are 2.8 and 3.2 nM respectively for human D2 and D3 and > 1000 nM for human D1, D4 and D5 receptors. Shows selectivity for presynaptic dopamine autoreceptors at low doses and blocks postsynaptic D2/D3 receptors at higher doses. Preferentially interacts with limbic D2-like receptors in vivo. Atypical antipsychotic/antischizophrenic agent with limited extrapyrimidal side effects and a profile distinct from that of haloperidol and remoxipride.
Purity: >98 %
在线咨询 联系方式 二维码

服务热线

021-60498804

扫一扫,关注我们