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/ Products Classification 点击展开+Cat. Number | 287080621940714 |
Chemical Name | AM 281 |
CAS Number | [202463-68-1] |
Mol. Formula | C21H19Cl2IN4O2 |
Mol. Weight | 557.22 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | 1-(2,4-Dichlorophenyl)-5-(4-iodophe nyl)-4-methyl-N-4-morpholinyl-1H-pyrazole-3-carbox amide |
Solubility | Soluble to 100 mM in DMSO |
Storage condition | Desiccate at +4°C |
References | Potent, selective CB1 cannabinoid receptor antagonist/inverse agonist (Ki values are 12 and 4200 nM for CB1 and CB2 receptors respectively). Increases locomotor activity following systemic administration in vivo. Analog of SR141716A (Ki = 14 nM). Purity: >99 % |