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Cat. Number
284869150776378
Chemical Name
BIO 1211
CAS Number
[187735-94-0]
Mol. Formula
C36H48N6O9
Mol. Weight
708.8
Qty 1
1mg
Storage condition
Store at -20°C
References
Selective, high affinity α4β1 (Very Late Antigen 4; VLA-4) inhibitor; displays 200-fold selectivity for the activated form of α4β1 (KD = 70 pM; IC50 = 0.004 μM). Selective for α4β1 over a range of other integrins (IC50 >100 μM for α1β1, α5β1 and α6β1).
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