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| Cat. Number | 283495105016077 |
| Chemical Name | CP 154526 |
| CAS Number | [157286-86-7] |
| Mol. Formula | C23H32N4.HCl |
| Mol. Weight | 400.99 |
| Qty 1 |
10mg |
| Qty 2 | 50mg |
| Synonym | N-Butyl-N-ethyl-2,5-dimethyl-7-(2,4 ,6-trimethylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-a mine hydrochloride |
| Solubility | Soluble to 50 mM in DMSO and to 50 mM in ethanol |
| Storage condition | Desiccate at +4°C |
| References | Selective, non-peptide CRF1 receptor antagonist (Ki values are 2.7 and > 10000 nM for CRF1 and CRF2 receptors respectively). Blocks CRF-induced adenylate cyclase activation (Ki = 3.7 nM) and attenuates activation of the HPA axis by CRF. Displays anxiolytic-like activity in the rat elevated plus-maze test; brain penetrant. Purity: >99 % |
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