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/ Products Classification 点击展开+Cat. Number | 279185692745961 |
Chemical Name | Dihydroergotoxine mesylate |
CAS Number | [8067-24-1] |
Qty 1 |
100mg |
Solubility | Soluble in ethanol |
Storage condition | Store at RT |
References | A complex of closely related alkaloid salts. Binds with high affinity to the GABAA receptor Cl- channel, producing an allosteric interaction with the benzodiazepine site. Also interacts with central dopaminergic, serotonergic and adrenergic (α1) receptors. Displays antiproliferative activity in vitro (IC50 = 18 - 38 μM in prostate cancer cells) and exhibits cognition-enhancing, anticonvulsant and sedative activity in vivo. Orally active. |