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Cat. Number
Exendin-4
Chemical Name
Exendin-4
CAS Number
[141758-74-9]
Mol. Formula
C184H282N50O60S
Mol. Weight
4186.61
Qty 1
1mg
Storage condition
Desiccate at -20°C
References
High affinity glucagon-like peptide 1 (GLP-1) receptor agonist (Kd = 136 pM); originally isolated from Heloderma suspectum venom. Potently induces cAMP formation without stimulating amylase release in pancreatic acini. Potentiates glucose-induced insulin secretion in isolated rat islets. Protects against glutamate-induced neurotoxicity.
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