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/ Products Classification 点击展开+Cat. Number | Gavestinel |
Chemical Name | Gavestinel |
CAS Number | [153436-22-7] |
Mol. Formula | C18H11Cl2N2O3Na |
Mol. Weight | 397.19 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | 4,6-Dichloro-3-[(1E)-3-oxo-3-(pheny lamino)-1-propenyl]-1H-indole-2-carboxylic acid sodium salt |
Solubility | Soluble to 40 mM in DMSO |
Storage condition | Desiccate at RT |
References | Highly potent and selective non-competitive antagonist acting at the strychnine-insensitive glycine binding site of the NMDA receptor-channel complex (Kd = 0.8 nM). Displays > 1000-fold selectivity over NMDA, AMPA and kainate binding sites. Orally bioavailable and active in vivo. Purity: >98 % |