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| Cat. Number | threo Ifenprodil hemitartrate |
| Chemical Name | threo Ifenprodil hemitartrate |
| CAS Number | [74991-34-7] |
| Mol. Formula | C21H27NO2.½C4H6O6 |
| Mol. Weight | 400.49 |
| Qty 1 |
10mg |
| Qty 2 | 50mg |
| Synonym | (1S*,2S*)-threo-2-(4-Benzylpiperidi no)-1-(4-hydroxyphenyl)-1-propanol hemitartrate |
| Solubility | Soluble to 25 mM in water and to 100 mM in DMSO |
| Storage condition | Store at RT |
| References | Potent σ receptor agonist (Ki values are 59.1 and 2 nM for σ1 and σ2 receptors respectively) and NR2B subunit-selective NMDA receptor antagonist (IC50 values are 0.22 and 324.8 μM at NR2B and NR2A respectively). Displays ~8-fold reduced affinity at α-adrenoceptors compared to Ifenprodil (Cat.No. 0545). Inhibits the hERG potassium channel (IC50 = 88 nM) and exhibits antiarrhythmic activity in vivo. |
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