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| Cat. Number | J 104129 fumarate |
| Chemical Name | J 104129 fumarate |
| CAS Number | [244277-89-2] |
| Mol. Formula | C24H36N2O2.C4H4O4 |
| Mol. Weight | 500.63 |
| Qty 1 |
10mg |
| Synonym | (αR)-α-Cyclopentyl-α-hydroxy-N-[1-(4-m ethyl-3-pentenyl)-4-piperidinyl]benzeneacetamide fumarate |
| Solubility | Soluble to 100 mM in DMSO and to 50 mM in ethanol |
| Storage condition | Store at +4°C |
| References | Potent M3 muscarinic receptor antagonist that displays ~ 120-fold selectivity over M2 receptors (Ki values are 4.2, 19 and 490 nM for human M3, M1 and M2 receptors respectively). Exhibits > 250-fold bronchial selectivity; inhibits ACh-induced bronchoconstriction but not ACh-induced bradycardia (KB values are 3.3 and 170 nM for rat trachea M3 and rat right atria M2 receptors respectively). Purity: >99 % |
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