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/ Products Classification 点击展开+Cat. Number | MRS 2279 |
Chemical Name | MRS 2279 |
CAS Number | [367909-40-8] |
Mol. Formula | C13H18ClN5O8P2.2NH3 |
Mol. Weight | 503.78 |
Qty 1 |
1mg |
Synonym | (1R*,2S*)-4-[2-Chloro-6-(methylamin o)-9H-purin-9-yl]-2-(phosphonooxy)bicyclo[3.1.0]he xane-1-methanol dihydrogen phosphate ester diammonium salt |
Solubility | Soluble to 100 mM in water |
Storage condition | Desiccate at -20°C |
References | Selective, high affinity competitive antagonist of the P2Y1 receptor (Ki = 2.5 nM; IC50 = 51.6 nM). Fails to block nucleotide signaling at most other P2Y receptors (P2Y2, P2Y4, P2Y6, P2Y11 and P2Y12) and potently inhibits ADP-induced aggregation of human blood platelets in vitro (pKB = 8.05). Purity: >98 % |