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| Cat. Number | Naloxone benzoylhydrazone |
| Chemical Name | Naloxone benzoylhydrazone |
| CAS Number | [119630-94-3] |
| Mol. Formula | C26H27N3O4 |
| Mol. Weight | 445.52 |
| Qty 1 |
10mg |
| Qty 2 | 50mg |
| Synonym | [(5α)-4,5-Epoxy-3,14-dihydroxy-17-(2 -propenyl)morphinan-6-ylidene] benzoic acid hydrazide |
| Solubility | Soluble to 50 mM in DMSO |
| Storage condition | Desiccate at +4°C |
| References | Mixed opioid receptor agonist/antagonist. Acts as a potent and full agonist at κ, a partial agonist at μ and δ opioid receptors (pEC50 values are 9.45, 8.74 and 8.61 in a cAMP assay, 9.70, 8.59 and 8.49 in a [35S]GTPγS binding assay respectively). Fails to exert agonist effects at NOP receptors and antagonizes agonist-induced NOP activation. Stimulates κ-, μ- and δ-mediated analgesia and blocks NOP-induced supraspinal nociception. Purity: >99 % |
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