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/ Products Classification 点击展开+Cat. Number | PK 44 phosphate |
Chemical Name | PK 44 phosphate |
CAS Number | [1017682-65-3] |
Mol. Formula | C17H16F5N7O.H3PO4 |
Mol. Weight | 527.34 |
Qty 1 |
10mg |
Synonym | (3R)-3-Amino-4-(6,7-difluoro-1H-ind azol-3-yl)-1-[5,6-dihydro-3-(trifluoromethyl)-1,2, 4-triazolo[4,3-a]pyrazin-7(8H)-yl]-1-butanone phosphate |
Solubility | Soluble to 100 mM in water and to 100 mM in DMSO |
Storage condition | Store at -20°C |
References | Potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50 = 15.8 nM). Displays >1000-fold selectivity for DPP-IV over DPP-8 and DPP-9. Improves glucose tolerance in a mouse oral glucose tolerance assay. Purity: >98 % |