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/ Products Classification 点击展开+Cat. Number | R-96544 hydrochloride |
Chemical Name | R-96544 hydrochloride |
CAS Number | [167144-79-8] |
Mol. Formula | C22H29NO3.HCl |
Mol. Weight | 391.94 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | (2R,4R)-5-[2-[2-[2-(3-Methoxyphenyl )ethyl]phenoxy]ethyl]-1-methyl-3-pyrrolidinol hydrochloride |
Solubility | Soluble to 100 mM in water and to 100 mM in DMSO |
Storage condition | Store at RT |
References | Potent, selective 5-HT2 receptor antagonist; displays some selectivity for 5-HT2A receptors (Ki = 1.6 nM). IC50 values are 2.2, 310, 2400, 3700, > 5000 and > 5000 nM for 5-HT2, α1-adrenergic, D2 dopamine, 5-HT1, 5-HT3 and β-adrenergic receptors respectively. Inhibits 5-HT-induced platelet aggregation and pressor responses in vivo. Purity: >99 % |