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/ Products Classification 点击展开+Cat. Number | Tiagabine hydrochloride |
Chemical Name | Tiagabine hydrochloride |
CAS Number | [145821-59-6] |
Mol. Formula | C20H25NO2S2.HCl |
Mol. Weight | 412.01 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | (3R)-1-[4,4-Bis(3-methyl-2-thienyl) -3-butenyl]-3-piperidinecarboxylic acid hydrochloride |
Solubility | Soluble to 50 mM in water and to 100 mM in DMSO |
Storage condition | Desiccate at RT |
References | GABA uptake inhibitor (IC50 = 67 nM in vivo). Exhibits high affinity and selectivity for the GAT-1 GABA transporter. Anticonvulsant; also attenuates established dynorphin-induced allodynia in a mouse model after systemic administration. Purity: >99 % |