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| Cat. Number | UBP 302 |
| Chemical Name | UBP 302 |
| Mol. Formula | C15H15N3O6 |
| Mol. Weight | 333.3 |
| Qty 1 |
10mg |
| Qty 2 | 50mg |
| Synonym | (S)-1-(2-Amino-2-carboxyethyl)-3-(2 -carboxybenzyl)pyrimidine-2,4-dione |
| Solubility | Soluble to 25 mM in 1eq. NaOH and to 50 mM in DMSO |
| Storage condition | Store at RT |
| References | Selective and potent GLUK5 (GluR5)-subunit containing kainate receptor antagonist (apparent KD = 402 nM); active enantiomer of UBP 296 (Cat. No. 2078). Displays ~ 260-fold selectivity over AMPA receptors. UBP 296 displays ~ 90-fold selectivity over recombinant human GLUK6- and GLUK2-containing kainate receptors, has little or no action at NMDA or group I mGlu receptors and selectively blocks kainate receptor-mediated LTP induction in rat hippocampal mossy fibres. Purity: >98 % |
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