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| Cat. Number | WIN 55,212-3 mesylate |
| Chemical Name | WIN 55,212-3 mesylate |
| CAS Number | [131543-25-4] |
| Mol. Formula | C27H26N2O3.CH3SO3H |
| Mol. Weight | 522.61 |
| Synonym | [(3S)-2,3-Dihydro-5-methyl-3-(4-mor pholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6- yl]-1-naphthalenyl-methanone monomethanesulfonate |
| Solubility | Soluble to 100 mM in DMSO |
| Storage condition | Store at +4°C |
| References | Novel, low potency CB2 receptor silent antagonist and CB1 receptor partial inverse agonist. Competitively antagonizes effects of CP 55,940 (pA2 = 6.1) and SR 144528 (pEC50 = 5.3) at CB2 receptors and acts as a partial inverse agonist at CB1 receptors (pIC50 = 5.5). Displays modest activity at human melatonin MT1 and muscarinic M4 receptors, but is selective over several other GPCRs. Purity: >98 % |
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