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/ Products Classification 点击展开+Cat. Number | Zamifenacin fumarate |
Chemical Name | Zamifenacin fumarate |
CAS Number | [127308-98-9] |
Mol. Formula | C27H29NO3.C4H4O4 |
Mol. Weight | 531.6 |
Qty 1 |
10mg |
Qty 2 | 50mg |
Synonym | (3R)-1-[2-(1-,3-Benzodioxol-5-yl)et hyl]-3-(diphenylmethoxy)piperidine fumarate |
Solubility | Soluble to 100 mM in DMSO and to 25 mM in ethanol |
Storage condition | Desiccate at +4°C |
References | Selective M3 muscarinic receptor antagonist (pKi values are 8.52, 7.93, 7.90 and 7.78 for M3, M2, M1 and M4 receptors respectively). Displays higher affinity at ileal M3 receptors (pKi = 9.3) compared to oesophageal and tracheal M3 receptors (pKi values are 8.8 and 8.2 respectively). Inhibits gastrointestinal motility in vivo in the absence of cardiovascular effects. Purity: >99 % |
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